Triazolam Pharmacology

Triazolam

About Triazolam
Short acting Benzodiazepine derivative, Hypnotic ,amnesic,anxiolytic, sedative, anticonvulsant, muscle relaxant.
Mechanism of Action of Triazolam
Triazolam mainly acts on Limbic system and ascending reticular formation in the CNS and binds to the BZD receptor. The binding will facilitates GABA mediated chloride channel opening and produce hyperpolarisation. This will produce an increase in the concentration of the inhibitory neurotransmitter GABA and chloride ions and decreases firing rate of neuron. These in turn alters normal functions of the body.
Pharmacokinets of Triazolam
Absorption: It is well absorbed after oral administration. Distribution: It is distributed widely in the body in protein bound form. Metabolism: It undergoes metabolism in the liver. Excretion: Metabolites are excreted mainly in the urine.
Onset of Action for Triazolam
15 - 20 minute
Duration of Action for Triazolam
N/A
Half Life of Triazolam
1.5 - 5.5 hour
Side Effects of Triazolam
1.Drowsiness
2.Headache
3.Dizziness
4.Nervousness
5.Light-headedness
6.Coordination disorders
7.Ataxia
8.Nausea
9.Vomiting
Contra-indications of Triazolam
Hypersensitivity to Triazolam and other Benzodiazepines
Special Precautions while taking Triazolam
1.Renal impairment
2.Hepatic impairment
3.Pulmonary insufficiency
4.Sleep apnea
5.Mental depression
6.Suicidal tendencies
7.Drug abuse
Pregnancy Related Information
contraindicated
Old Age Related Information
Use with caution
Breast Feeding Related Information
contraindicated
Children Related Information
contraindicated
Indications for Triazolam
Insomnia
Interactions for Triazolam
N/A
Typical Dosage for Triazolam
Oral
Adult: 0.125 - 0.25mg at bed time. Maximum dose: 0.5mg
Schedule of Triazolam
N/A
Storage Requirements for Triazolam
The drug should be kept at 15 - 30 degree C in a tightly closed container.
Effects of Missed Dosage of Triazolam
Take the missed dose as soon as noticed and if it is the time for next dose then skip the missed dose.
Effects of Overdose of Triazolam
Give support and symptomatic treatment. Flumazenil can be given as antagonist. Hypotension can be treated with vasopressors.If the patient is conscious induce emesis followed by charcoal administration

Home Delivery for Triazolam in Your City

Medicine India is just a publishing medium for medicine related information and does not provide services or sales of medicines including triazolam.

However, we do publish a comprehensive directory of Pharmacies, Chemists and Druggists in cities all over India. You can use this directory to find the medicine stores in your city (or area) that provide home delivery services for triazolam and other medicines and health products. Home delivery services for triazolam may be free or they may cost you depending on the pharmacy and the minimum order requirements. It would be best to get this clarified while placing the order.

Please be aware that you should take triazolam only if a doctor has recommended or prescribed it. Some or all pharmacies who provide a home delivery service for medicines might insist on a prescription for triazolam before they complete the sale. You can get this information while placing the order for triazolam with the pharmacy.

Triazolam is a generic medicine name and there are several brands available for it. Some of the brands for triazolam might be better known than triazolam itself. If the pharmacy that's willing to deliver medicines to your home doesn't have triazolam in stock, you can ask for one of the branded alternatives for triazolam.